GPR6 inverse agonist 2

SKU: orb3210829

Description

GPR6inverse agonist 2 (Compound 575) is a selective inverse agonist of GPR6, displaying IC50 values of 50 of 21.71 μM for hERG. GPR6inverse agonist 2 is applicable in research on movement disorders such as Parkinson's disease.

Key Properties

• CAS Number: 3029155-57-2
• MW: 523.58
• Formula: C₂₇H₃₁F₂N₇O₂
• SMILES: C(C)N1C=C(C=2C(=NC3=C(N2)C=NC([C@@H](C(C)(C)O)O)=C3)N4CCN(CC5=C(F)C=C(F)C=C5)CC4)C=N1
• Target: GPCR

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

GPCR