GPR4 antagonist 1

SKU: orb1709554

Description

GPR4 antagonist 1 is a potent small molecule inhibitor of the G protein-coupled receptor GPR4, exhibiting an IC50 of 189 nM. This compound is a valuable research tool for investigating the role of GPR4 in physiological and pathological processes, such as inflammation and cancer, in both cellular and animal models.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1197879-16-5
• MW: 431.62
• Formula: C₂₇H₃₇N₅
• SMILES: CCc1nc2c(C)cc(C)nc2n1Cc1ccc(\C=C\CN2CCN(CC2)C(C)C)cc1
• Target: GPCR

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

57970302