GPBAR1-IN-3

SKU: orb1689170

Description

GPBAR1-IN-3 (Compound 14) is a dual-function small molecule, acting as a selective GPBAR1 agonist (EC50 = 0.17 µM) and a CysLT1R antagonist. This profile supports its use in research exploring metabolic and inflammatory pathways, applicable in both in vitro and in vivo experimental models.

Research Area

Pharmacology & Drug Discovery, Signal Transduction

Key Properties

• CAS Number: 2760546-05-0
• MW: 321.41
• Formula: C₂₁H₂₃NO₂
• SMILES: C(OC1=CC(OCC(CC)C)=CC=C1)C2=NC3=C(C=C2)C=CC=C3
• Target: GPCR19,Others,Leukotriene Receptor

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

168277662