GP 1a

SKU: orb1690050

Description

GP 1a is a potent and selective CB2 receptor agonist (EC50=7.1 nM) with demonstrated efficacy in cellular assays, including cAMP inhibition and ERK1/2 phosphorylation. It exhibits anti-inflammatory and anti-fibrotic properties, promoting epithelial regeneration, which supports its research application in models of skin wound healing and tissue repair.

Research Area

Cell Biology, Pharmacology & Drug Discovery, Signal Transduction

Key Properties

• CAS Number: 511532-96-0
• MW: 441.35
• Purity: 99.96% (May vary between batches)
• Formula: C₂₃H₂₂Cl₂N₄O
• SMILES: C(NN1CCCCC1)(=O)C=2C3=C(N(N2)C4=C(Cl)C=C(Cl)C=C4)C=5C(C3)=CC(C)=CC5
• Target: ERK,Cannabinoid Receptor
• Solubility: Ethanol:90 mg/mL (203.92 mM);DMSO:90 mg/mL (203.92 mM)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

GP 1a, CB2, Cannabinoid Receptor, CannabinoidReceptor, PERK

Compound Identifiers

PubChem CID

10252734