GNE-781

• Catalog Number: orb1308265
• Category: Small Molecules
• Description: GNE-781
• CAS Number: [1936422-33-1]
• Purity: 98.73%
• MW: 525.59
• SMILES: CNC(=O)N1CCc2c(C1)c(nn2C1CCOCC1)N1CCCc2cc(-c3cnn(C)c3)c(cc12)C(F)F
• Formula: C₂₇H₃₃F₂N₇O₂
• Biological Activity: GNE-781 is a highly potent and selective inhibitor of CBP (IC50: 0.94 nM in TR-FRET assay). GNE-781 also inhibits BRET and BRD4(1) (IC50s: 6.2 nM and 5100 nM, respectively).
• Storage: -20°C
• Note: For research use only
• Expiration Date: 12 months from date of receipt.