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GNE-617

SKU: orb1222733

Description

GNE-617 is a potent nicotinamide phosphoribosyltransferase (NAMPT) inhibitor with IC50 value of 5nM. Prolonged inhibition of nicotinamide phosphoribosyltransferase (NAMPT) is a strategy for targeting cancer metabolism.

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Key Properties

CAS Number1362154-70-8
MW427.43
Purity>98% (HPLC)
FormulaC21H15F2N3O3S
SMILESC1=CC(=CC=C1CNC(=O)C2=CN3C=CN=C3C=C2)S(=O)(=O)C4=CC(=CC(=C4)F)F
TargetJNK
SolubilityDMSO : ≥ 42.85 mg/mL; 100.25 mM

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

GNE-617 | GNE 617 | GNE617

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Protocol Information

GNE-617 (orb1222733)

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% DMSO +
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% Tween 80 +
%

Available Sizes

Select a size below

2 mg
$ 90.00
5 mg
$ 130.00
10 mg
$ 190.00
25 mg
$ 330.00
50 mg
$ 500.00
100 mg
$ 730.00
500 mg
$ 1,550.00