GAC Inhibitor 968

SKU: orb1303506

Description

Glutaminase C-IN-1 (Compound 968) is a cell-permeable, allosteric inhibitor of glutaminase C (GAC). It is widely used in cancer metabolism research to study glutamine dependency in vitro and has been shown to inhibit tumor growth in various xenograft models in vivo.

Research Area

Protein Biochemistry

Key Properties

• CAS Number: 311795-38-7
• MW: 475.4
• Purity: >98%
• Formula: C₂₇H₂₇BrN₂O
• SMILES: CN(C)C1=C(Br)C=C(C=C1)C1NC2=CC=C3C=CC=CC3=C2C2=C1C(=O)CC(C)(C)C2
• Target: Glutaminase
• Solubility: Soluble in DMSO (up to (11 mg/ml); or ethanol (up to 1 mg/ml, warm)

Storage & Handling

• Storage: RT
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Inhibitor, Glutaminase, Glutaminase C allosteric, Glutaminase C IN 1, Glutaminase CIN1, Glutaminase C-IN-1, Glutaminase Inhibitor Compound 968, inhibit, Compound 968, Compound-968, Compound968

Compound Identifiers

PubChem CID

3099980