Gemfibrozil 1-O-β-glucuronide

SKU: orb1992846

Description

Gemfibrozil 1-O-β-Glucuronide is the major glucuronide metabolite of the drug gemfibrozil and acts as a potent, competitive inhibitor of the cytochrome P450 enzyme CYP2C8 (IC₅₀ = 4.07 µM). It is a valuable research tool for studying drug-drug interactions and CYP2C8 metabolism in both in vitro and in vivo experimental models.

Research Area

Metabolism Research, Molecular Biology

Key Properties

• CAS Number: 91683-38-4
• MW: 426.46
• Formula: C₂₁H₃₀O₉
• SMILES: Cc1ccc(C)c(OCCCC(C)(C)C(=O)O[C@@H]2O[C@@H]([C@@H](O)[C@H](O)[C@H]2O)C(O)=O)c1
• Target: PPAR,Others,Drug Metabolite,Cytochromes P450

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

88127