G-Protein antagonist peptide acetate

SKU: orb1296452

Description

G-Protein antagonist peptide acetate is a substance P-derived peptide that competitively inhibits G-protein coupling to specific receptors. It blocks Gi/Go activation by M2 mAChR and Gs activation by beta-adrenergic receptors in reconstituted systems, as measured by GTPase assays. This tool is used in vitro to study G-protein-mediated signaling pathways and receptor-effector interactions.

Research Area

Pharmacology & Drug Discovery

Key Properties

• Target: Adrenergic Receptor
• MW: 1153.33
• Purity: 98.06% (May vary between batches)
• Formula: C₅₉H₆₈N₁₂O₁₁S
• SMILES: CSCC[C@@H](C(N)=O)NC([C@@H](CC1=CNC2=CC=CC=C12)NC([C@H](NC([C@H](CC3=CC=CC=C3)NC([C@H](NC([C@H](CCC(N)=O)NC([C@H]4NC(CC4)=O)=O)=O)CC5=CNC6=CC=CC=C56)=O)=O)CC7=CNC8=CC=CC=C78)=O)=O.CC(O)=O

Storage & Handling

• Storage: store at low temperature,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

AdrenergicReceptor, Adrenergic Receptor, GProtein antagonist peptide acetate, G-Protein antagonist peptide Acetate, G Protein antagonist peptide acetate

Compound Identifiers

PubChem CID

168013632