FL104

SKU: orb1700597

Description

FL104 is a potent small-molecule agonist for the urotensin II receptor (UT receptor), exhibiting a pEC50 of 7.11. This compound is a valuable research tool for investigating the UT system in cardiovascular and renal pathophysiology, suitable for both in vitro and in vivo experimental models.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 885672-81-1
• MW: 392.92
• Purity: 99.46% (May vary between batches)
• Formula: C₂₄H₂₅ClN₂O
• SMILES: C(NC(=O)C1=CC=C(C=C1)C2=CC=CC=C2)(CCN(C)C)C3=CC=C(Cl)C=C3
• Target: Others,GPCR
• Solubility: DMSO:9 mg/mL (22.91 mM)

Bioactivity

• Target IC50:
  UTII receptor:7.11 (pEC50)
• In Vitro:
  FL104 were tested for the ability to stimulate the human urotensin II receptor using a functional R-SATTM assay, pEC50= 7.11.

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

FL 104, FL104, FL-104, Urotensin Receptor (GPR14)

Compound Identifiers

PubChem CID

11663047