(E/Z)-GSK5182?

SKU: orb1220077

Description

(E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active estrogen-related receptor γ (ERRγ) inverse agonist(IC50 of 79 nM),and also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma.

Key Properties

• Target: Estrogen Receptor/ERR
• Molecular Weight: 417.54
• Purity: >98% (HPLC)
• CAS Number: ——
• Formula: C₂₇H₃₁NO₃
• SMILES: CN(C)CCOC1=CC=C(C=C1)C(=C(CCCO)C1=CC=CC=C1)C1=CC=C(O)C=C1

Storage & Handling

• Storage: Storage temperature: -20°C. Stability: ≥ 2 years
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

GSK5182(Z/E)

Quick Database Links

Gene Symbol

Estrogen Receptor/ERR