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ET receptor antagonist 1

SKU: orb2277844

Description

ET Receptor Antagonist 1 (compound 16h) is a potent, orally bioavailable agent with an IC50 of 0.18 nM. It is a valuable research tool for pulmonary arterial hypertension (PAH), having shown in vivo efficacy in ameliorating monocrotaline-induced PAH in rat models.

Research Area

Metabolism Research

Images & Validation

Key Properties

MW459.52
FormulaC21H25N5O5S
TargetEstrogen Receptor/ERR

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Protocol Information

ET receptor antagonist 1 (orb2277844)

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Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

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