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ET receptor antagonist 1

ET receptor antagonist 1

Catalog Number: orb2277844

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Catalog Numberorb2277844
CategorySmall Molecules
DescriptionET Receptor Antagonist 1 (compound 16h), with an IC50 value of 0.18 nM, is an orally active agent that can be utilized for pulmonary arterial hypertension (PAH) research. It has demonstrated efficacy in mitigating monocrotaline-induced PAH in a rat model [1].
Purity98.00%
MW459.52
FormulaC21H25N5O5S
Biological ActivityET Receptor Antagonist 1 (compound 16h), with an IC50 value of 0.18 nM, is an orally active agent that can be utilized for pulmonary arterial hypertension (PAH) research. It has demonstrated efficacy in mitigating monocrotaline-induced PAH in a rat model [1].
Storage-20°C
NoteFor research use only
Expiration Date12 months from date of receipt.
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