BQ-788

SKU: orb181359

Description

BQ-788 sodium salt is a potent, selective ETB receptor antagonist (IC50 = 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells); poorly inhibited the binding to ET A receptors in human neuroblastoma cell line SK-N-MC cells (IC(50), 1300 nM).

Key Properties

• CAS Number: 156161-89-6
• MW: 663.779880046844
• Purity: >98%
• Formula: C₃₄H₅₀N₅NAO₇
• SMILES: [Na+].CCCC[C@@H](N(C([C@@H](NC(N1[C@H](C)CCC[C@@H]1C)=O)CC(C)(C)C)=O)C([C@@H](CC1=CN(C(OC)=O)C2=CC=CC=C12)N)=O)C([O-])=O

Storage & Handling

• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Chemical structure of BQ-788