EST64454 Maleic acid salt

SKU: orb1298198

Description

EST64454 Maleic acid salt is the salt form of EST64454, a highly soluble σ1 receptor antagonist developed as a clinical candidate for pain treatment. Its application in research includes investigating σ1 receptor pharmacology in both in vitro binding assays and in vivo models of neuropathic and inflammatory pain.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 2088272-67-5
• MW: 480.46
• Purity: 98.71% (May vary between batches)
• Formula: C₂₂H₂₆F₂N₄O₆
• SMILES: CC(N1CCN(CCOCC2=NN(C3=CC=C(F)C(F)=C3)C=C2)CC1)=O.O=C(O)/C=C\C(O)=O
• Target: Sigma receptor,Others
• Solubility: DMSO:60 mg/mL (124.88 mM)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

EST64454 Maleic acid, EST64454 Maleic acid salt, EST-64454 Maleic acid salt

Compound Identifiers

PubChem CID

135316606