ERK5-IN-5

SKU: orb1944732

Description

ERK5-IN-5 is a potent and selective inhibitor of extracellular signal-regulated kinase 5 (ERK5) with demonstrated anticancer activity. It inhibits the proliferation of A549 non-small cell lung cancer cells in vitro and has shown potential anticonvulsant effects in preclinical research models.

Research Area

Signal Transduction, Stem Cell & Developmental Biology

Key Properties

• CAS Number: 2318792-30-0
• MW: 337.8
• Purity: 99.89% (May vary between batches)
• Formula: C₁₉H₁₆ClN₃O
• SMILES: O=C(C1=CC=C(Cl)C=C1)N2CC=C(C3=CNC=4N=CC=CC43)CC2
• Target: ERK
• Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (5.92 mM);DMSO:55 mg/mL (162.82 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

ERK5, ERK5IN5

Compound Identifiers

PubChem CID

52403715