ERK5-IN-4

SKU: orb1688409

Description

ERK5-IN-4 (compound 34b) is a potent and selective ERK5 inhibitor, demonstrating activity against both full-length and truncated ERK5 (ΔTAD) in cellular assays with IC50 values of 77 nM and 300 nM, respectively. This tool compound is used in vitro to investigate the role of ERK5 signaling in cancer, inflammation, and cardiovascular disease research.

Research Area

Signal Transduction, Stem Cell & Developmental Biology

Key Properties

• CAS Number: 1888305-17-6
• MW: 381.19
• Formula: C₁₆H₁₁Cl₂FN₄O₂
• SMILES: C(=O)(C=1C=C(C(NC=2C=NN(C)C2)=O)NC1)C3=C(F)C(Cl)=CC=C3Cl
• Target: ERK,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

118959090