Enzastaurin HCl

• Catalog Number: orb1737641
• Category: Small Molecules
• Description: Enzastaurin HCl
• Purity: 98.00%
• MW: 552.08
• Biological Activity: Enzastaurin HCl, also known as DB-102 and LY317615, is a synthetic macrocyclic bisindolemaleimide with potential antineoplastic activity. Binding to the ATP-binding site, Enzastaurin HCl selectively inhibits protein kinase C beta, an enzyme involved in the induction of vascular endothelial growth factor (VEGF)-stimulated neo-angiogenesis. This agent may decrease tumor blood supply and so tumor burden.
• CAS Number: 359017-79-1
• Formula: C₃₂H₃₀ClN₅O₂
• SMILES: Cl.Cn1cc(C2=C(C(=O)NC2=O)c2cn(C3CCN(Cc4ccccn4)CC3)c3ccccc23)c2ccccc12
• Storage: -20°C
• Note: For research use only