Enzastaurin 2HCl

• Catalog Number: orb1740126
• Category: Small Molecules
• Description: Enzastaurin 2HCl
• Purity: 98.00%
• MW: 588.53
• Biological Activity: Enzastaurin 2HCl, also known as DB-102 and LY317615, is a synthetic macrocyclic bisindolemaleimide with potential antineoplastic activity. Binding to the ATP-binding site, Enzastaurin 2HCl selectively inhibits protein kinase C beta, an enzyme involved in the induction of vascular endothelial growth factor (VEGF)-stimulated neo-angiogenesis. This agent may decrease tumor blood supply and so tumor burden.
• CAS Number: 365253-37-8
• Formula: C₃₂H₃₁Cl₂N₅O₂
• SMILES: O=C1C(C=2C=3C(N(C2)C4CCN(CC5=CC=CC=N5)CC4)=CC=CC3)=C(C(=O)N1)C=6C=7C(N(C)C6)=CC=CC7.Cl.Cl
• Storage: -20°C
• Note: For research use only