Endoxifen HCl

SKU: orb1222919

Description

Z-Endoxifen HCl is an estrogen receptor alpha (ERalpha) ligand, potent antiestrogen, and metabolite of tamoxifen. Z-endoxifen is the most potent of the metabolites of tamoxifen, and has the potential to be more effective than tamoxifen because it bypasses potential drug resistance mechanisms attributable to patient variability in the expression of the hepatic microsomal enzyme CYP2D6.

Key Properties

• CAS Number: 1032008-74-4
• MW: 409.95
• Purity: >98% (HPLC)
• Formula: C₂₅H₂₈ClNO₂
• SMILES: CC/C(=C(\c1ccc(cc1)O)/c1ccc(cc1)OCCNC)/c1ccccc1.Cl
• Target: Sodium Channel
• Solubility: DMSO : 12.5 mg/mL 30.49 mM; H2O : < 0.1 mg/mL

Storage & Handling

• Storage: Storage temperature: -20°C. Stability: ≥ 2 years
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Z-Endoxifen HCl | Z Endoxifen HCl | ZEndoxifen Hydrochloride

Quick Database Links

Gene Symbol

Sodium Channel