Enciprazine dihydrochloride

SKU: orb3211235

Description

Enciprazine dihydrochloride is an orally active non-benzodiazepine anxiolytic agent. It functions as a 5-HT1A receptor (5-HT1AR) agonist and an α1-adrenergic receptor antagonist. This compound induces changes in drug-induced EEG by decreasing the average power of δ and θ waves while increasing the average power of α and fast β waves. Enciprazine dihydrochloride exhibits anti-aggressive activity with only mild sedative and ataxic effects. It modulates plasma corticosterone levels and activates the hypothalamic-pituitary-adrenal axis. Enciprazine dihydrochloride is applicable in studies related to anxiety disorders, generalized anxiety syndrome, and psychotic conditions.

Key Properties

• CAS Number: 68576-88-5
• MW: 505.43
• Formula: C₂₃H₃₄Cl₂N₂O₆
• SMILES: OC(CN1CCN(CC1)C2=C(OC)C=CC=C2)COC3=CC(OC)=C(OC)C(OC)=C3.Cl.Cl
• Target: Adrenergic Receptor,5-HT Receptor

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

Adrenergic Receptor,5-HT Receptor