EGFR/HER2/CDK9-IN-2

SKU: orb1686686

Description

EGFR/HER2/CDK9-IN-2 is a potent triple inhibitor targeting EGFR, HER2, and CDK9 with respective IC50 values of 145.35, 129.07, and 117.13 nM. It demonstrates significant antitumor activity in biochemical and cellular assays, supporting its use as a research tool in oncology for studying kinase-driven cancer pathways.

Research Area

Cardiovascular Research, Cell Biology, Epigenetics & Chromatin; Cell Biology, Signal Transduction

Key Properties

• CAS Number: 1180924-34-8
• MW: 496.56
• Formula: C₂₃H₂₀N₄O₅S₂
• SMILES: C(CC1=CC=C(S(N)(=O)=O)C=C1)N2C(SCC3=CC=C(N(=O)=O)C=C3)=NC=4C(C2=O)=CC=CC4
• Target: CDK,Others,EGFR

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

36982442