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EGFR-IN-42

EGFR-IN-42

Catalog Number: orb1982923

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Catalog Numberorb1982923
CategorySmall Molecules
DescriptionEGFR-IN-42 (Compound 17b), a potent EGFR inhibitor, demonstrates single-digit nanomolar activity by covalently linking tamoxifen or endoxifen with gefitinib, retaining both ER antagonist activity and EGFR inhibition, resulting in superior anti-cancer activity [1].
Purity98.00%
MW846.43
FormulaC49H53ClFN5O5
Biological ActivityEGFR-IN-42 (Compound 17b), a potent EGFR inhibitor, demonstrates single-digit nanomolar activity by covalently linking tamoxifen or endoxifen with gefitinib, retaining both ER antagonist activity and EGFR inhibition, resulting in superior anti-cancer activity [1].
Storage-20°C
NoteFor research use only
Expiration Date12 months from date of receipt.