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DSP-1053

SKU: orb1709824

Description

DSP-1053 is a potent serotonin transporter (SERT) inhibitor with high affinity (Ki=1.02 nM) and also acts as a partial agonist at the 5-HT1A receptor (Ki=5.05 nM). This pharmacological profile makes it a useful research tool for investigating serotonin neurotransmission in models of depression, anxiety, and related CNS disorders in both in vitro and in vivo studies.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number1176326-76-3
MW502.44
FormulaC26H32BrNO4
SMILESCOCCOc1cc(CC2CCN(CCc3ccc4OCCC(=O)c4c3)CC2)ccc1Br
Target5-HT Receptor,Serotonin Transporter,Others

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Key Properties

No computed properties available.

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Protocol Information

DSP-1053 (orb1709824)

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(Recommended: An additional animal making an allowance for loss during the experiment)

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