Difelikefalin HCl

SKU: orb1739943

Description

Difelikefalin HCl is a potent and selective κ-opioid receptor (KOR) agonist, as demonstrated by its low-nanomolar EC₅₀ in cellular assays. It exhibits in vivo efficacy, reducing pain-related writhing and KOR antagonist-induced scratching in mice. This compound is a valuable research tool for studying KOR pharmacology in neurobiology, pruritus, and pain research contexts.

Key Properties

• CAS Number: 2711717-77-8
• MW: 789.237
• Formula: C₃₆H₅₃N₇O₆.xHCl
• SMILES: C([C@H](NC([C@H](NC([C@@H](CC1=CC=CC=C1)NC([C@@H](CC2=CC=CC=C2)N)=O)=O)CC(C)C)=O)CCCCN)(=O)N3CCC(C(O)=O)(N)CC3.Cl
• Target: Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

172652788