Queen's Award Received in 2021 ISO 9001 Certified Delivered over 1,000,000 bio-reagents to life science researchers Trusted by Life Science Communities
Cart summary

You have no items in your shopping cart.

CRT0066101

SKU: orb2566590

Description

CRT0066101 is a potent, orally bioavailable small-molecule inhibitor of PKD isoforms (PKD1/2/3 IC₅₀ 1-2.5 nM) with additional activity against PIM2. It exhibits anticancer properties and has been utilized in research exploring oncology, cell signaling, and in vitro mechanistic studies as well as in vivo tumor models.

Research Area

Cell Biology, Epigenetics & Chromatin, Metabolism Research, Signal Transduction

Images & Validation

Key Properties

CAS Number956123-34-5
MW338.41
FormulaC18H22N6O
SMILESOC=1C(=CC(=CC1)C2=CN(C)N=C2)C=3N=C(NC[C@@H](CC)N)C=CN3
TargetSerine/threonin kinase,Pim

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Similar Products

  • CRT0066101 dihydrochloride [orb1296201]

    99.85% (May vary between batches)

    1883545-60-5

    411.33

    C18H22N6O.2HCl

    50 mg, 5 mg, 10 mg, 25 mg, 1 mg, 1 ml x 10 mM (in DMSO), 100 mg
  • CRT0066101 hydrochloride [orb2283813]

    1781742-22-0

    374.87

    C18H23ClN6O

    10 mg, 5 mg, 1 mg
  • PKD-IN-1 dihydrochloride (956121-30-5 free base) [orb1298493]

    99.92% (May vary between batches)

    2308510-39-4

    415.75

    C18H21Cl3N4O

    5 mg, 10 mg, 25 mg, 50 mg, 100 mg, 1 ml x 10 mM (in DMSO), 2 mg
  • CRT0066101 [orb1217428]

    >98% (HPLC)

    956121-30-5

    342.82

    C18H19ClN4O

    5 mg, 10 mg, 25 mg, 50 mg, 100 mg, 200 mg, 500 mg, 1 g
  • CRT0066101 dihydrochloride(956121-30-5 free base) [orb1218367]

    >98% (HPLC)

    2308510-39-4

    415.74

    C18H21N4OCl3

    5 mg, 10 mg, 25 mg, 50 mg, 100 mg, 200 mg, 500 mg, 1 g
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

Protocol Information