CPI-1328

SKU: orb1690927

Description

CPI-1328 is a highly potent, femtomolar-range inhibitor of EZH2, with a Ki of 63 fM. This small molecule is a valuable research tool for investigating epigenetic mechanisms in oncology, supporting both in vitro biochemical assays and in vivo cancer model studies.

Research Area

Epigenetics & Chromatin

Key Properties

• CAS Number: 2390367-27-6
• MW: 546.12
• Formula: C₂₈H₃₆ClN₃O₄S
• SMILES: [H][C@@]1(CC[C@@H](CC1)N(C)C)[C@]1(C)Oc2c(O1)c(Cl)c1CCN(Cc3c(SC)cc(C)[nH]c3=O)C(=O)c1c2C |wU:4.7,1.0,wD:10.11,1.10,(9.17,1.25,;8.85,-.26,;8.53,-1.77,;9.67,-2.8,;11.14,-2.32,;11.46,-.81,;10.31,.22,;12.28,-3.35,;13.75,-2.88,;11.96,-4.86,;7.7,.77,;8.85,1.8,;6.8,2.02,;5.33,1.54,;5.33,,;6.8,-.48,;4,-.77,;4,-2.31,;2.67,,;1.33,-.77,;;,1.54,;-1.33,2.31,;-2.67,1.54,;-2.67,,;-1.33,-.77,;-1.33,-2.31,;-4,-.77,;-5.33,,;-6.67,-.77,;-5.33,1.54,;-4,2.31,;-4,3.85,;1.33,2.31,;1.33,3.85,;2.67,1.54,;4,2.31,;4,3.85,)|
• Target: Others,Histone Methyltransferase

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

153367388