Conteltinib tetrahydrochloride

SKU: orb2945499

Description

Conteltinib tetrahydrochloride (CT-707 tetrahydrochloride) is a potent small molecule inhibitor targeting FAK, ALK, and Pyk2, with an IC50 of 1.6 nM against FAK. Research demonstrates its synergistic antitumor activity with Cabozantinib in preclinical models, supporting its investigation in oncology, particularly for cancers involving these kinase pathways.

Research Area

Cardiovascular Research, Signal Transduction

Key Properties

• MW: 781.667
• Formula: C₃₂H₄₉Cl₄N₉O₃S
• SMILES: CC(C)NS(=O)(=O)C1=CC=CC=C1NC2=NC(=NC3=C2CCN3)NC4=C(C=C(C=C4)N5CCC(CC5)N6CCN(CC6)C)OC.Cl.Cl.Cl.Cl
• Target: FAK

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

172676750