CLP-3094

SKU: orb1298305

Description

CLP-3094

Research Area

Immunology & Inflammation

Key Properties

• CAS Number: 312749-73-8
• MW: 304.8
• Purity: >98%
• Formula: C₁₅H₁₃ClN₂OS
• SMILES: ClC1=CC=C(OCCSC2=NC3=CC=CC=C3N2)C=C1
• Target: GPCR
• Solubility: Soluble in DMSO (up to 45 mg/ml)

Bioactivity

• Target IC50:
  BF3 (Androgen receptor):4 μM
• In Vivo:
  I.p. administration of 30, 100 mg/kg CLP-3094 daily from Day 0 to Day 11 consistently displayed significantly lower severity of arthritis scores than vehicle-treated mice and reduced the arthritis scores dose-dependently, by not much..
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Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

prostate, resistance, CLP 3094, CLP3094, CLP-3094, antiandrogens, Androgen Receptor, AndrogenReceptor, cancer, 2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE, inhibit, LNCaP, Inhibitor

Compound Identifiers

PubChem CID

1736098