Cloperidone

SKU: orb2564685

Description

Cloperidone is a CYP2C9 inhibitor (IC50 = 17.7 µM) that demonstrates cytotoxic effects in vitro, reducing HepG2 cell viability to 60% at 10 µM. This small molecule is a useful research tool for studying CYP2C9-mediated metabolism and drug interactions in biochemical and cellular assays.

Research Area

Metabolism Research

Key Properties

• CAS Number: 4052-13-5
• MW: 398.89
• Formula: C₂₁H₂₃ClN₄O₂
• SMILES: O=C1NC=2C=CC=CC2C(=O)N1CCCN3CCN(C=4C=CC=C(Cl)C4)CC3
• Target: Cytochromes P450

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

10675