CJ 033466

SKU: orb1305855

Description

CJ 033466 is a potent and selective 5-HT4 receptor partial agonist (EC50 = 9 nM). This compound exhibits gastroprokinetic activity and is utilized in gastrointestinal motility research, including in vitro receptor studies and in vivo models for functional analysis.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 519148-48-2
• MW: 377.91
• Purity: 99.72%
• Formula: C₁₉H₂₈ClN₅O
• SMILES: CC(C)CN1CCC(CNC(=O)c2cc(Cl)c(N)n3cc(C)nc23)CC1
• Target: 5-HT Receptor
• Solubility: Ethanol:< 37.79 mg/mL;DMSO:10 mg/mL (26.46 mM)

Bioactivity

• Target IC50:
  5-HT4 receptor:9 nM (EC50)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Serotonin Receptor, Inhibitor, gastrointestinal dysfunction, gastroprokinetic, inhibit, CJ 033466, CJ033466, CJ-033466, 5HT Receptor, 5-HT Receptor, 5HTReceptor, 5-hydroxytryptamine Receptor, 5-HT4

Compound Identifiers

PubChem CID

10429706