Cilengitide TFA

SKU: orb1908980

Description

Cilengitide is a potent integrin inhibitor for αvβ3 receptor and αvβ5 receptor with IC50 of 4.1 nM and 79 nM in cell-free assays, respectively; ~10-fold selectivity against gpIIbIIIa. Phase 2.

Research Area

Cell Biology, Signal Transduction

Key Properties

• CAS Number: 199807-35-7
• MW: 702.68
• Formula: C₂₉H₄₁F₃N₈O₉
• SMILES: OC(=O)C(F)(F)F.CC(C)[C@@H]1N(C)C(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](CC(O)=O)NC(=O)CNC(=O)[C@H](CCCNC(N)=N)NC1=O
• Target: Autophagy,Integrin

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

129626550