CBP/p300-IN-3

SKU: orb1309287

Description

CBP/p300-IN-3 is a potent small molecule inhibitor targeting the histone acetyltransferase activity of p300 and CBP. It is a valuable chemical probe for epigenetic research, used in vitro and in vivo to study the roles of these enzymes in cancer, cellular differentiation, and other disease contexts.

Research Area

Epigenetics & Chromatin, Signal Transduction

Key Properties

• CAS Number: 2299226-01-8
• MW: 431.53
• Purity: 99.14% (May vary between batches)
• Formula: C₂₄H₂₉N₇O
• SMILES: CCN(CC)c1ccc(cn1)-c1nc2cc(ccc2n1Cc1ccn(CC)n1)C(=O)NC
• Target: Histone Acetyltransferase
• Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:5 mg/mL (11.59 mM);DMSO:250 mg/mL (579.33 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

P300/CBP-IN-3, inhibit, Inhibitor, HistoneAcetyltransferase, histone acetyltransferase, Histone Acetyltransferase, HATs, HAT, CBP/p300IN3, CBP/p-300-IN-3, CBP/p300-IN-3, CBP/p300 IN 3

Compound Identifiers

PubChem CID

138466007