CBP/p300-IN-18

SKU: orb1687323

Description

CBP/p300-IN-18 is a potent and selective dual inhibitor of the histone acetyltransferases EP300 and CBP, with IC50 values of 0.056 µM and 0.46 µM against H3K27 acetylation, respectively. This small molecule is a valuable chemical probe for epigenetic research, enabling the investigation of p300/CBP HAT function in cancer and other disease models both in vitro and in vivo.

Research Area

Epigenetics & Chromatin, Signal Transduction

Key Properties

• MW: 450.51
• Formula: C₂₅H₂₇FN₄O₃
• Target: Others,Histone Acetyltransferase

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

Others,Histone Acetyltransferase