Cavα2δ1&NET-IN-3

SKU: orb1744726

Description

Cavα2δ1&NET-IN-3 (example 216) is a dual-target small molecule inhibitor of the voltage-gated calcium channel α2δ-1 subunit and the norepinephrine transporter (NET), with Ki values of approximately 100 nM and 500 nM, respectively. This compound is a useful research tool for investigating pain signaling and sympathetic nervous system function in both cellular and animal models.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 2143584-82-9
• MW: 466.6
• Formula: C₂₄H₃₀N₆O₂S
• SMILES: O=C1C=2C(=NC(NCC)=NC2)N(C)CCN1C3=CC(O[C@@H](CCNC)C4=CC=CS4)=CC=C3
• Target: Calcium Channel,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

132088914