Carazolol

SKU: orb1224608

Description

Carazolol is a high affinityantagonist/partial inverse agonist (also referred to as abeta blocker) of the β-adrenergic receptor.(In Vivo):Carazolol (0.01 mg/kg; i.m.; once) shows no significant side effects.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 57775-29-8
• MW: 298.38
• Purity: >98% (HPLC)
• Formula: C₁₈H₂₂N₂O₂
• SMILES: OC(CNC(C)C)COC1=CC=CC(N2)=C1C3=C2C=CC=C3
• Target: Adrenergic Receptor
• Solubility: Soluble in DMSO

Bioactivity

• In Vivo:
  Carazolol (0.01 mg/kg; i. m. ; once) shows no significant side effects. Animal model: Kivircik sheeps, 25-45 kg, nonpregnant. Dosage: 0.01 mg/kg. Administration: Intramuscular injection, once. Result: Urea, creatinin, ALT, ALP, GGT, LDH, Ca, P, T. Protein, Mg, Cu levels in blood serum parameters were found to be in normal level however serum Fe, Zn levels were decreased.

Storage & Handling

• Storage: Storage temperature: -20°C. Stability: ≥ 2 years
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

BM 51052 | (±)-Carazolol

Quick Database Links

Gene Symbol

Adrenergic Receptor