Bremelanotide Acetate

SKU: orb1299663

Description

Bremelanotide Acetate is supplied for research use only and is intended for laboratory research involving animal models. Biorbyt supplies these products exclusively to research institutions and commercial laboratories.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1607799-13-2
• MW: 1085.22
• Purity: 96.72%
• Formula: C₅₂H₇₂N₁₄O₁₂
• SMILES: CC(O)=O.[H][C@]1(CCCCNC(=O)C[C@H](NC(=O)[C@H](CCCC)NC(C)=O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@]([H])(Cc2ccccc2)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1)C(O)=O
• Target: Melanocortin Receptor
• Solubility: DMSO:122.5 mg/mL (112.88 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (1.84 mM)

Bioactivity

• In Vivo:
  Treatment with Bremelanotide (100 or 200 μg/kg) significantly increased proceptive solicitations in females primed with E+Por E alone (E+O) in bilevel chambers
• Animal Research:
  Bremelanotide(PT-141), a cyclic heptapeptide melanocortin analogue (Palatin Technologies, Cranbury, NJ), was dissolved in saline to obtain doses of 50, 100, and 200 μg/kg/ml, and injected s.c. 5 min before each behavioral test. An equal volume of saline was administered to control animals.

Storage & Handling

• Storage: keep away from moisture,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

MelanocortinReceptor, Melanocortin Receptor, Bremelanotide Acetate, PT141, PT-141, PT141 Acetate, PT-141 Acetate, PT 141, PT 141 Acetate

Compound Identifiers

PubChem CID

91971505