BRD7116

SKU: orb1305608

Description

BRD7116 is a competitive inhibitor of bacterial DNA gyrase. This small molecule exhibits cell-non-autonomous activity against leukemia, making it a candidate for research in oncology and microbiology. It is suitable for both in vitro enzymatic assays and in vivo leukemia model studies.

Research Area

Infectious Disease & Virology, Molecular Biology

Key Properties

• CAS Number: 329059-55-4
• MW: 496.66
• Purity: 99.91%
• Formula: C₂₈H₃₆N₂O₄S
• SMILES: CC1(C)C(C(=O)NC2C=CC(=CC2=S(=O)=O)c2ccc(NC(=O)C3C(C)(C)C3(C)C)cc2)C1(C)C
• Target: DNA gyrase,Antibacterial
• Solubility: DMSO:4.97 mg/mL (10.01 mM)

Bioactivity

• Target IC50:
  DNA gyrase:200 nM (EC50)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

inhibit, Inhibitor, Bacterial, BRD 7716, BRD 7116, BRD7116, BRD-7116, BRD7716, BRD-7716, DNA gyrase, DNAgyrase

Compound Identifiers

PubChem CID

91895228