BRD-IN-3

SKU: orb1710210

Description

BRD-IN-3 is a potent and selective small molecule inhibitor of the PCAF bromodomain with an IC50 of 7 nM, also demonstrating activity against GCN5 and FALZ. This compound is a valuable chemical probe for epigenetic research, enabling the study of bromodomain function in both cellular assays and in vivo models of cancer and inflammation.

Research Area

Epigenetics & Chromatin

Key Properties

• CAS Number: 2351938-32-2
• MW: 395.45
• Formula: C₂₁H₂₅N₅O₃
• SMILES: N([C@@H]1C[C@@H](CN(C)C1)C=2C=C3C(=CC2)OCCO3)C4=NC5=C(C(=O)N4C)NC=C5
• Target: Epigenetic Reader Domain,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

138105961