Bragsin1

SKU: orb1707515

Description

Bragsin1 is a potent, selective, and noncompetitive inhibitor of the ArfGEF BRAG2, blocking Arf GTPase activation with an IC50 of 3 µM. This small molecule exhibits anti-cancer activity and is a valuable chemical probe for studying Arf-dependent signaling pathways in cancer cell proliferation and invasion, both in vitro and in vivo.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 369631-68-5
• MW: 273.16
• Formula: C₁₁H₆F₃NO₄
• SMILES: Cc1ccc2oc(cc(=O)c2c1[N+]([O-])=O)C(F)(F)F
• Target: GTPase,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

740511