BigLEN (mouse) acetate

SKU: orb1296376

Description

BigLEN (mouse) acetate is a highly potent and selective small molecule agonist for the orphan receptor GPR171, exhibiting a dissociation constant (Kd) of approximately 0.5 nM. This tool compound is valuable for investigating GPR171 signaling in both in vitro cellular assays and in vivo models related to metabolic regulation and immune function.

Research Area

Metabolism Research, Neuroscience, Pharmacology & Drug Discovery

Key Properties

• Target: GPCR
• MW: 1816.07
• Purity: >99.99% (May vary between batches)
• Formula: C₈₀H₁₃₄N₂₄O₂₄
• SMILES: O=C(O)[C@H]1N(C([C@H]2N(C([C@H](CC(C)C)NC([C@H](CC(C)C)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](C)NC([C@H]3N(C([C@H](C)NC([C@H](CCC(N)=O)NC([C@H]4N(C([C@H](CO)NC([C@H]5N(C([C@H](CC(N)=O)NC([C@H](CCC(O)=O)NC([C@H](CC(C)C)N)=O)=O)=O)CCC5)=O)=O)CCC4)=O)=O)=O)CCC3)=O)=O)=O)=O)=O)=O)CCC2)=O)CCC1.CC(O)=O

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

501036-69-7, 501036-69-7 Free base, BigLEN, BigLEN Acetate, BigLEN (mouse) acetate, BigLEN (mouse) acetate (501036-69-7 Free base), GPR171

Compound Identifiers

PubChem CID

163285800