BETd-246

SKU: orb1707569

Description

BETd-246 is a potent inhibitor of second-generation and PROTAC-based BET bromodomain proteins, demonstrating antitumor activity. It is a valuable research tool for studying BET function in oncology, with applications in both in vitro biochemical assays and in vivo cancer models.

Research Area

Epigenetics & Chromatin, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 2140289-17-2
• MW: 946.02
• Formula: C₄₈H₅₅N₁₁O₁₀
• SMILES: O=C(NCCCOCCOCCOCCCNC1=CC=CC=2C(=O)N(C(=O)C12)C3C(=O)NC(=O)CC3)C4=NC=5NC=6C=C(C(OC)=CC6C5C(=N4)NC7=CC(=NN7CC)C8CC8)C=9C(=NOC9C)C
• Target: PROTACs,Epigenetic Reader Domain

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

131698640