BET-IN-16

SKU: orb1944392

Description

BET-IN-16 (Comp I) is a potent BET bromodomain inhibitor that suppresses prostate cancer cell proliferation, exhibiting IC50 values of 0.043 μM in LNCaP and 0.034 μM in 22Rv1 cells. This small molecule is a valuable research tool for investigating BET protein function in oncology, with applications in both in vitro mechanistic studies and in vivo cancer model research.

Research Area

Epigenetics & Chromatin

Key Properties

• CAS Number: 2089390-09-8
• MW: 515.56
• Formula: C₃₁H₂₅N₅O₃
• SMILES: C(C)(N1C=2C(C(=C1)C3=CC=C(C(O)=O)C=C3)=NC=C(C2)C=4C(C)=NOC4C)(C5=CC=CC=N5)C6=CC=CC=N6
• Target: Epigenetic Reader Domain

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

126689208