AZ-GHS-38

SKU: orb3174700

Description

AZ-GHS-38 (compound 38) is an orally active inverse agonist of the growth hormone secretagogue receptor (GHS-R1a) that can cross the blood-brain barrier, with an IC50 of 6.7 nM. It has been shown to acutely reduce food intake in wild-type mice and may be used for anti-obesity research.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1143021-16-2
• MW: 578.1
• Formula: C₂₅H₂₈ClN₅O₅S₂
• SMILES: O=C(NC(=O)C1=CC(=CC=C1Cl)N2CCOCC2)NC3=NC=4C=CC(=CC4S3)S(=O)(=O)C5CCN(C)CC5
• Target: GHSR

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

GHSR