AS2521780

SKU: orb1707639

Description

AS2521780 is a potent and selective small molecule inhibitor of protein kinase C-theta (PKCθ), exhibiting an IC50 of 0.48 nM. This compound is a valuable research tool for studying T-cell activation and immune signaling pathways in both cellular and animal models of inflammation and autoimmunity.

Research Area

Epigenetics & Chromatin, Signal Transduction

Key Properties

• CAS Number: 1214726-89-2
• MW: 547.76
• Formula: C₃₀H₄₁N₇OS
• SMILES: C(NC=1C(C#N)=CN=C(NCC2=C(SC)N=CC=C2)N1)C34C[C@@]5([C@@H](NC[C@@H]6CC[C@@H](O)CC6)[C@](C3)(CC(C4)C5)[H])[H]
• Target: PKC

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

58324913