Aplithianines A

SKU: orb1941786

Description

Aplithianines A is a potent, ATP-competitive inhibitor of protein kinase A, showing an IC50 of 84 nM against wild-type PKA and 1 μM for J-PKAcα. This small molecule is a valuable research tool for in vitro studies targeting PKA-mediated signaling pathways in cancer and cellular regulation.

Research Area

Signal Transduction

Key Properties

• CAS Number: 3027425-38-0
• MW: 299.36
• Formula: C₁₃H₁₃N₇S
• SMILES: N=1C=C(C=2SCCN(C2)C3=NC=NC=4N=CNC43)N(C1)C
• Target: PKA

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

PKA