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APJ receptor agonist 1
Catalog Number: orb1691035
| Catalog Number | orb1691035 |
|---|---|
| Category | Small Molecules |
| Description | APJ receptor agonist 1 |
| Purity | 98.00% |
| MW | 524.02 |
| Biological Activity | APJ receptor agonist 1, a potent biphenyl acid derivative, acts as an agonist (EC50 of 0.093 nM and 0.12 nM for human and rat APJ receptors, respectively) for the APJ receptor (APJ-R). It exhibits significant in vitro potency towards apelin-13, the endogenous peptidic ligand for the APJ receptor. APJ receptor agonist 1 holds promise for heart failure research. |
| CAS Number | 2287153-38-0 |
| Formula | C31H26ClN3O3 |
| SMILES | CCCC(NC(=O)c1ccc(c(c1)C(O)=O)-c1c(Cl)cccc1-c1nc2ccccc2[nH]1)c1ccccc1 |
| Storage | -20°C |
| Note | For research use only |
[Pyr1]-Apelin-13 [orb1219858]
> 98% (HPLC)
217082-60-5
1533.8
C69H108N22O16S
1 g, 500 mg, 200 mg, 50 mg, 100 mg, 25 mg, 5 mg, 10 mg
