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APD668

SKU: orb1306510

Description

APD668

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number832714-46-2
MW477.51
Purity99.97%
FormulaC21H24FN5O5S
SMILESCC(C)OC(=O)N1CCC(CC1)Oc1ncnc2n(ncc12)-c1ccc(cc1F)S(C)(=O)=O
TargetPotassium Channel,Cytochromes P450,GPCR
SolubilityDMSO:45 mg/mL (94.24 mM)

Bioactivity

Target IC50
CYP2C9:0.1 μM (Ki)|ERG channel (human):3 μM|GPR119 (human):2.7 nM (EC50)|GPR119 (rat):33 nM (EC50)

Storage & Handling

StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

G-protein, G Protein-Coupled Receptor 119, GPR119, KcsA, Inhibitor, inhibit, APD 668, APD668, APD-668, coupled, Cytochrome P450, CYPs, CYP2C9, diabetes, steatohepatitis, PotassiumChannel, Potassium Channel

Similar Products

  • APD 668 [orb1223917]

    >98%(HPLC)

    832714-46-2

    477.5

    C21H24FN5O5S

    1 g, 500 mg, 200 mg, 10 mg, 2 mg, 25 mg, 50 mg, 100 mg, 5 mg
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Key Properties

No computed properties available.

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Protocol Information

APD668 (orb1306510)

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% DMSO +
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% Tween 80 +
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Available Sizes

Select a size below

1 mg
$ 90.00
5 mg
$ 150.00
1 ml x 10 mM (in DMSO)
$ 160.00
10 mg
$ 210.00
25 mg
$ 340.00
50 mg
$ 530.00
100 mg
$ 730.00
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