Anticancer agent 258

SKU: orb2814596

Description

Anticanceragent 258 is a potent imidazotriazole-based modulator of Nurr1 (EC50=63 nM in N2A cells) and Nur77 (IC50=0.1 pM in HEK293 cells). This small molecule is a valuable research tool for investigating nuclear receptor function in cancer biology, metabolic disease, and neurological disorder models, both in vitro and in vivo.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 2891984-12-4
• MW: 310.3
• Formula: C₁₇H₁₂F₂N₄
• SMILES: FC=1C=CC(=CC1)C=2N=C3N(N2)C=C(C=4C=CC=C(F)C4)N3C
• Target: Orphan Receptor,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

166473718