Anpirtoline hydrochloride

SKU: orb1704683

Description

Anpirtoline hydrochloride is a dual-action small molecule, functioning as a 5-HT1B receptor agonist and 5-HT3 receptor antagonist. It exhibits analgesic and antidepressant properties in preclinical studies and is utilized in research on pain, depression, and movement disorders, including in vivo models of neuropathic pain.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 99201-87-3
• MW: 265.20
• Purity: >99.99% (May vary between batches)
• Formula: C₁₀H₁₄Cl₂N₂S
• SMILES: Cl.ClC=1N=C(SC2CCNCC2)C=CC1
• Target: 5-HT Receptor
• Solubility: DMSO:10 mg/mL (37.71 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (3.77 mM);H2O:10 mg/mL (37.71 mM)

Storage & Handling

• Storage: keep away from moisture | Pure form: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

5-HT3, 5HT Receptor, 5-HT1B, 5HTReceptor, D-16949 hydrochloride

Compound Identifiers

PubChem CID

6917943