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Acefylline

SKU: orb1306111

Description

Acefylline is a xanthine-class adenosine receptor antagonist with stimulant properties. It is used in research to study adenosine signaling and is formulated with diphenhydramine in preparations like Etanautine to counteract its stimulant effects. Its applications include in vitro receptor binding assays and investigations into respiratory and neurological pathways.

Research Area

Cell Biology, Epigenetics & Chromatin, Metabolism Research, Molecular Biology, Neuroscience, Pharmacology & Drug Discovery, Signal Transduction

Images & Validation

Key Properties

CAS Number652-37-9
MW238.2
Purity99.57% (May vary between batches)
FormulaC9H10N4O4
SMILESCN1C2=C(N(CC(O)=O)C=N2)C(=O)N(C)C1=O
TargetHDAC,PKA,TNF,PAD,Adenosine Receptor,PDE
Solubility10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (8.4 mM);DMSO:50 mg/mL (209.91 mM)

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

Carboxymethyltheophylline, AdenosineReceptor, Adenosine Receptor, Acefylline, A2, A1, A3, acetyloxytheophylline, PDE4, Inhibitor, inhibit, HDAC2, TNF-α, Protein Arginine Deiminase, P1 receptor, Peptidylarginine Deiminase, Theophylline-7-acetic acid, Theophyllineacetic acid, PKA, Phosphodiesterase (PDE), phosphodiesterase

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Quality Guarantee

Quality Guarantee

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Key Properties

No computed properties available.

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Acefylline (orb1306111)

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% DMSO +
%+
% Tween 80 +
%

Available Sizes

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50 mg
$ 80.00
100 mg
$ 90.00
1 ml x 10 mM (in DMSO)
$ 100.00
DispatchUsually dispatched within 3-5 working days
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